SCHEMBL624331

SCHEMBL624331

B(Oc1ccc(OC2CCCCC2)nc1)Oc1ccc(OC2CCCCC2)nc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LOX P28300 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
ACACB O00763 7/20 0.39
PDGFRB P09619 3/20 0.38
PDGFRA P16234 3/20 0.38
ACACA Q13085 1/20 0.37
ABL1 P00519 1/20 0.36
HRH3 Q9Y5N1 3/20 0.36
NAMPT P43490 1/20 0.34
TDO2 P48775 1/20 0.34
KCNH2 Q12809 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017157 0.84 PIK3CA (0.37) ACACBHRH3NAMPTTDO2
SCHEMBL30748869 0.75 LOX (0.46) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL15147591 0.75 PDGFRB (0.44) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL1644324 0.75 LOX (0.43) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL16839481 0.75 FPR2 (0.46) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL3651197 0.75 LOX (0.46) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL625001 0.75 DGAT1 (0.46) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL16839464 0.75 TDO2 (0.44) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL16924081 0.75 LOX (0.43) LOXLOXL2ACACBPDGFRBPDGFRA
SCHEMBL16839487 0.73 KDM4E (0.45) LOXLOXL2ACACBPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2603513-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2013-06-19 EP disclosed
WO-2012020848-A1 HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-02-16 WO disclosed