SCHEMBL624417

SCHEMBL624417

C1=C2Oc3ccccc3N=C2c2ccccc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
HRH4 Q9H3N8 4/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
HRH2 P25021 2/20 0.32
HRH1 P35367 2/20 0.32
HTR6 P50406 2/20 0.32
KCNK2 O95069 1/20 0.32
ADRB2 P07550 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14164372 0.84 HTR6 (0.37) CYP1A2CYP2D6HRH4KDM4ENPC1
SCHEMBL29413193 0.79 MEN1 (0.32) CYP1A2CYP2D6HRH4KDM4ENPC1
SCHEMBL214039 0.73 IDO1 (0.38) HRH4KDM4EALDH1A1LMNAMAPT
SCHEMBL30518953 0.67 DRD2 (0.38) HRH4KDM4EALDH1A1LMNAHRH2
SCHEMBL29438383 0.65 MAOA (0.45) KDM4ENPC1ALDH1A1LMNAGAA
SCHEMBL667761 0.65 MAOA (0.45) KDM4ENPC1ALDH1A1LMNAGAA
SCHEMBL15549945 0.65 KDM4E (0.36) CYP1A2CYP2D6HRH4KDM4ENPC1
SCHEMBL29870245 0.65 CYP1A2 (0.41) CYP1A2CYP2D6HRH4KDM4ENPC1
SCHEMBL5438463 0.63 HDAC3 (0.61) CYP1A2CYP2D6HRH4HDAC3HDAC1
SCHEMBL2059873 0.63 KDM4E (0.32) CYP1A2CYP2D6KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2591355-A2 IN VITRO POINT-OF-CARE SENSOR AND METHOD OF USE CASE WESTERN RESERVE UNIVERSITY (US) 2013-05-15 EP disclosed
WO-2012021239-A9 IN VITRO POINT-OF-CARE SENSOR AND METHOD OF USE CASE WESTERN RESERVE UNIVERSITY (US) 2012-05-31 WO disclosed
WO-2012021239-A2 IN VITRO POINT-OF-CARE SENSOR AND METHOD OF USE CASE WESTERN RESERVE UNIVERSITY (US) 2012-02-16 WO disclosed