SCHEMBL6244302

SCHEMBL6244302

Nc1nc(N2CCCC2)c(N)c(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2C9 P11712 1/20 0.42
NUDT1 P36639 1/20 0.42
LMNA P02545 2/20 0.41
CTSK P43235 2/20 0.41
HSD17B10 Q99714 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 4/20 0.41
ADORA2A P29274 3/20 0.41
HPGD P15428 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
SLC9A5 Q14940 2/20 0.41
PLAU P00749 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
MEN1 O00255 2/20 0.41
TP53 P04637 2/20 0.41
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28323735 0.74 LMNA (0.56) MAPTCYP1A2CYP2C19CYP2C9NUDT1
SCHEMBL17822435 0.72 CTSK (0.52) MAPTCYP1A2CYP2C19CYP2C9NUDT1
SCHEMBL17822445 0.70 LMNA (0.55) LMNACTSKHSD17B10ALDH1A1TSHR
SCHEMBL17822430 0.70 LMNA (0.55) LMNACTSKHSD17B10ALDH1A1TSHR
SCHEMBL9663929 0.69 LMNA (0.50) MAPTCYP1A2CYP2C19CYP2C9NUDT1
SCHEMBL12457406 0.69 ALDH1A1 (0.44) MAPTCYP1A2CYP2C19CYP2C9NUDT1
Hydrochloric Acid SCHEMBL17822431 0.68 LMNA (0.53) LMNACTSKHSD17B10ALDH1A1TSHR
SCHEMBL5774307 0.68 MEN1 (0.47) LMNACTSKHSD17B10MEN1KMT2A
Hydrochloric Acid SCHEMBL6250270 0.68 LMNA (0.49) MAPTCYP1A2CYP2C19CYP2C9NUDT1
SCHEMBL27741341 0.68 HSD17B10 (0.44) MAPTCYP1A2CYP2C19CYP2C9NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546129-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS ANTITUMOR AGENT Pharmacia Italia S.p.A. (IT) 2005-06-29 EP disclosed
WO-2004024711-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS ANTITUMOR AGENT PHARMACIA ITALIA S.P.A. (IT) 2004-03-25 WO disclosed