SCHEMBL6247334

SCHEMBL6247334

Fc1cc(-c2nc3ccccc3[nH]2)cc(F)c1F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 13/20 0.65
RAB9A P51151 13/20 0.65
KDM4E B2RXH2 12/20 0.65
SMN1; SMN2 Q16637 10/20 0.65
ALDH1A1 P00352 12/20 0.63
HPGD P15428 5/20 0.63
MAPT P10636 5/20 0.63
HSD17B10 Q99714 4/20 0.63
USP2 O75604 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
GAA P10253 1/20 0.62
PKM P14618 6/20 0.60
TP53 P04637 4/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
ABCB11 O95342 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
PKN1 Q16512 1/20 0.57
PKN2 Q16513 1/20 0.57
POLB P06746 3/20 0.56
GFER P55789 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12153689 0.85 NPC1 (0.77) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL3336689 0.85 NPC1 (0.68) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL15497747 0.83 NPC1 (0.74) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL6258373 0.81 NPC1 (0.69) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL3332901 0.80 NPC1 (0.66) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL27983509 0.79 ALDH1A1 (0.63) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL29386825 0.79 NPC1 (0.88) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL2178266 0.79 NPC1 (0.88) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL3337878 0.79 NPC1 (1.00) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL3417301 0.78 NPC1 (0.78) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551811-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS VANILLOID RECEPTOR LIGANDS Amgen Inc. (US) 2005-07-13 EP claimed
WO-2004035549-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS VANILLOID RECEPTOR LIGANDS AMGEN INC. (US) 2004-04-29 WO claimed