SCHEMBL6248381

SCHEMBL6248381

CC1(C)CNc2ccccc2C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
PDGFRA P16234 1/20 0.39
FER P16591 1/20 0.39
LTK P29376 1/20 0.39
CDK8 P49336 1/20 0.39
ACVR1 Q04771 1/20 0.39
LRRK2 Q5S007 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
KDM4E B2RXH2 3/20 0.38
HPGD P15428 3/20 0.38
PDK2 Q15119 1/20 0.37
PDK4 Q16654 1/20 0.37
GSK3B P49841 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
MAPT P10636 2/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579713 0.74 HTR2C (0.40) ALDH1A1MAOAMAOBSMN1; SMN2MAPT
SCHEMBL5260675 0.74 KDM4E (0.37) ALDH1A1MAOAMAOBPDGFRAFER
SCHEMBL2636968 0.72 MAPT (0.54) ALDH1A1CYP3A4MAPTTDP1POLB
SCHEMBL8577537 0.72 TDP2 (0.43) ALDH1A1KDM4EHPGDGSK3BMAPT
SCHEMBL3432668 0.72 LIG1 (0.39) ALDH1A1MAOAMAOBPDGFRAFER
SCHEMBL1031209 0.71 PDK2 (0.42) PDK2PDK4POLBBRD4
SCHEMBL29384370 0.71 PDK2 (0.42) PDK2PDK4POLBBRD4
SCHEMBL25631719 0.70 L3MBTL1 (0.48) ALDH1A1MAOAKDM4EGSK3BSMN1; SMN2
Hydrochloric Acid SCHEMBL2482151 0.69 PDK2 (0.41) ALDH1A1KDM4EHPGDPDK2PDK4
SCHEMBL13469502 0.69 ALDH1A1 (0.52) ALDH1A1MAOAMAOBPDGFRAFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583745-A1 1-PROPANOL AND 1-PROPYLAMINE DERIVATIVES AND THEIR USE AS GLUCOCORTICOID LIGANDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2005-10-12 EP claimed
WO-2004063163-A1 1-PROPANOL AND 1-PROPYLAMINE DERIVATIVES AND THEIR USE AS GLUCOCORTICOID LIGANDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-07-29 WO claimed