SCHEMBL624949

SCHEMBL624949

COc1cncc(-c2cnc3sc(N4CCC(C(=O)O)CC4)nn23)c1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FYN P06241 9/20 0.55
NEK2 P51955 3/20 0.46
KCNH2 Q12809 5/20 0.45
PIK3CA P42336 1/20 0.45
HASPIN Q8TF76 2/20 0.44
NR2F2 P24468 1/20 0.42
RAB9A P51151 1/20 0.42
KIT P10721 1/20 0.42
PIM1 P11309 1/20 0.42
FLT3 P36888 1/20 0.42
CDK7 P50613 1/20 0.42
PIM3 Q86V86 1/20 0.42
PIM2 Q9P1W9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625663 0.91 FYN (0.56) FYNKCNH2PIK3CAHASPINNR2F2
SCHEMBL624950 0.82 MAPT (0.56) NEK2
SCHEMBL626697 0.76 CYP11B2 (0.53) FYNPIK3CAHASPIN
SCHEMBL625664 0.74 MAPT (0.58)
SCHEMBL1945183 0.72 FYN (0.58) FYNPIK3CA
SCHEMBL18613694 0.71 FYN (1.00) FYNHASPIN
SCHEMBL1944166 0.70 FYN (0.81) FYNPIK3CAHASPIN
SCHEMBL1945181 0.70 FYN (0.87) FYNPIK3CA
SCHEMBL625746 0.70 PIK3CA (0.54) NEK2KCNH2PIK3CAHASPINKIT
SCHEMBL624430 0.69 FYN (0.72) FYNPIK3CAHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed