SCHEMBL626697

SCHEMBL626697

COc1cncc(-c2cnc3sc(N4CCCC4=O)nn23)c1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.53
CYP11B1 P15538 8/20 0.53
FYN P06241 9/20 0.50
PIK3CA P42336 1/20 0.48
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HASPIN Q8TF76 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626698 0.82 CYP11B2 (0.52) CYP11B2CYP11B1CYP1A2CYP3A4CYP2C9
SCHEMBL624949 0.76 FYN (0.55) FYNPIK3CAHASPIN
SCHEMBL625663 0.75 FYN (0.56) FYNPIK3CAHASPIN
SCHEMBL627766 0.72 L3MBTL1 (0.40)
SCHEMBL1762361 0.70 CYP11B1 (1.00) CYP11B2CYP11B1CYP1A2CYP3A4CYP2C9
SCHEMBL1945183 0.70 FYN (0.58) FYNPIK3CA
SCHEMBL1944166 0.69 FYN (0.81) FYNPIK3CAHASPIN
SCHEMBL532334 0.68 PIK3CA (0.64) FYNPIK3CA
SCHEMBL1945181 0.67 FYN (0.87) FYNPIK3CA
SCHEMBL624430 0.67 FYN (0.72) FYNPIK3CAHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed