SCHEMBL625663

SCHEMBL625663

COC(=O)C1CCN(c2nn3c(-c4cncc(OC)c4)cnc3s2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FYN P06241 8/20 0.56
PIK3CA P42336 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HASPIN Q8TF76 1/20 0.43
MAPT P10636 2/20 0.43
THRB P10828 1/20 0.43
KCNH2 Q12809 4/20 0.43
LMNA P02545 1/20 0.42
NR2F2 P24468 1/20 0.42
RAB9A P51151 1/20 0.42
GSK3B P49841 1/20 0.42
DYRK1A Q13627 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624949 0.91 FYN (0.55) FYNPIK3CAHASPINKCNH2NR2F2
SCHEMBL625664 0.83 MAPT (0.58) MAPTTHRB
SCHEMBL625746 0.79 PIK3CA (0.54) PIK3CAHASPINKCNH2
SCHEMBL627054 0.78 KDM4E (0.48) KDM4EMAPTTHRBLMNA
SCHEMBL626697 0.75 CYP11B2 (0.53) FYNPIK3CAHASPIN
SCHEMBL624950 0.74 MAPT (0.56) MAPTTHRB
SCHEMBL18613694 0.72 FYN (1.00) FYNHASPIN
SCHEMBL1945183 0.72 FYN (0.58) FYNPIK3CA
SCHEMBL1944166 0.71 FYN (0.81) FYNPIK3CAHASPIN
SCHEMBL1945181 0.71 FYN (0.87) FYNPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed