SCHEMBL625109

SCHEMBL625109

Cc1c(-c2cnc(N)c(C(F)(F)F)c2)nc2sc(NC3CCN(S(C)(=O)=O)CC3)nn12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.46
CCNE1 P24864 12/20 0.46
CCND1 P24385 12/20 0.41
CDK1 P06493 12/20 0.41
CDK4 P11802 11/20 0.41
CDK6 Q00534 8/20 0.41
CCNB1 P14635 8/20 0.41
CCND3 P30281 7/20 0.41
MAP3K12 Q12852 1/20 0.41
PIK3CA P42336 3/20 0.39
CCNT1 O60563 1/20 0.37
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37
CCNH P51946 1/20 0.37
MNAT1 P51948 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626189 0.91 MAP3K12 (0.42) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL625108 0.89 CDK2 (0.42) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL626206 0.86 PIK3CA (0.53) MAP3K12PIK3CA
SCHEMBL626188 0.86 MAP3K12 (0.41) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL626207 0.83 MAP3K12 (0.46) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL625753 0.78 PIK3CA (0.49) MAP3K12PIK3CA
SCHEMBL627467 0.76 HASPIN (0.43) MAP3K12PIK3CACCNT1
SCHEMBL627322 0.75 FYN (0.48) MAP3K12PIK3CA
SCHEMBL626795 0.75 PIK3CA (0.41) MAP3K12PIK3CA
SCHEMBL625754 0.74 MAP3K12 (0.40) MAP3K12PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed