SCHEMBL625754

SCHEMBL625754

CCCS(=O)(=O)N1CCC(Nc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 13/20 0.40
PIK3CA P42336 4/20 0.39
EPHX2 P34913 1/20 0.38
JAK1 P23458 1/20 0.36
NPY5R Q15761 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626207 0.90 MAP3K12 (0.46) MAP3K12PIK3CA
SCHEMBL624428 0.84 MAP3K12 (0.47) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL625301 0.82 MAP3K12 (0.44) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL627397 0.81 PIK3CA (0.49) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL625456 0.81 MAP3K12 (0.41) MAP3K12PIK3CA
SCHEMBL627328 0.81 PIK3CA (0.44) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL627440 0.81 FYN (0.45) MAP3K12PIK3CA
SCHEMBL625236 0.81 MAP3K12 (0.45) MAP3K12PIK3CA
SCHEMBL625128 0.80 CCNA2 (0.46) MAP3K12PIK3CAJAK1
SCHEMBL625636 0.80 MAP3K12 (0.44) MAP3K12PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed