SCHEMBL6251471

SCHEMBL6251471

CCS(=O)(=O)c1ccc(C2=C(c3ccc(OC)cc3)CCC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.72
PTGS1 P23219 8/20 0.72
SLC6A3 Q01959 1/20 0.50
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12883762 0.85 PKM (0.57) PTGS2PTGS1KDM4EALDH1A1MMP8
SCHEMBL213353 0.84 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6708168 0.83 PKM (0.64) ALDH1A1MMP8MMP13
SCHEMBL8651545 0.83 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8993420 0.81 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL7865484 0.81 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL8993482 0.79 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL2622585 0.79 PTGS2 (0.68) PTGS2PTGS1SLC6A3KDM4EALDH1A1
SCHEMBL8993358 0.76 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8993402 0.76 PTGS2 (0.74) PTGS2PTGS1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572239-A1 METHOD OF USING A COX-2 INHIBITOR AND A TOPOISOMERASE II INHIBITOR AS A COMBINATION THERAPY IN THE TREATMENT OF NEOPLASIA Pharmacia Corporation (US) 2005-09-14 EP disclosed
WO-2004058302-A1 METHOD OF USING A COX-2 INHIBITOR AND A TOPOISOMERASE II INHIBITOR AS A COMBINATION THERAPY IN THE TREATMENT OF NEOPLASIA PHARMACIA CORPORATION (US) 2004-07-15 WO disclosed