SCHEMBL6253671

SCHEMBL6253671

CC(C)c1cccc(Nc2ncco2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.44
BRAF P15056 6/20 0.43
RAF1 P04049 3/20 0.43
EGFR P00533 2/20 0.42
TNNI3K Q59H18 1/20 0.42
KIF11 P52732 1/20 0.39
ERBB2 P04626 1/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
JAK2 O60674 2/20 0.37
SYK P43405 1/20 0.37
FFAR2 O15552 1/20 0.36
ALOX5 P09917 1/20 0.36
AURKA O14965 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532117 0.76 EGFR (0.50) EGFRAURKA
SCHEMBL544111 0.76 MEN1 (0.50) EGFRERBB2SYKFADS1
SCHEMBL16740946 0.76 KIF11 (0.54) IDO1BRAFEGFRTNNI3KKIF11
SCHEMBL24943110 0.76 IDO1 (0.52) IDO1BRAFEGFRTNNI3KKIF11
SCHEMBL729232 0.75 FLT1 (0.46) AURKA
SCHEMBL6237657 0.74 AURKA (0.57) EGFRKIF11AURKA
SCHEMBL10094216 0.72 EGFR (0.50) IDO1BRAFEGFRTNNI3KKIF11
SCHEMBL544110 0.72 NPC1 (0.44) AURKA
SCHEMBL543837 0.72 HDAC3 (0.42)
SCHEMBL4934839 0.71 FADS1 (0.31) FADS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed