SCHEMBL6237657

SCHEMBL6237657

FC(F)(F)c1cccc(Nc2ncco2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.57
KIF11 P52732 1/20 0.55
IDH2 P48735 3/20 0.53
THRB P10828 1/20 0.50
PTK6 Q13882 1/20 0.49
LMNA P02545 3/20 0.49
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 1/20 0.49
GMNN O75496 1/20 0.49
TTR P02766 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
PKM P14618 1/20 0.49
NFKB1 P19838 1/20 0.49
UGT1A1 P22309 1/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
PMP22 Q01453 1/20 0.49
DHODH Q02127 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30041659 0.80 EPHX2 (0.48) DHODH
SCHEMBL4532117 0.78 EGFR (0.50) AURKAEGFRABCG2RAPGEF4
SCHEMBL544111 0.78 MEN1 (0.50) PTK6LMNAALDH1A1MEN1KMT2A
SCHEMBL394991 0.77 KIF11 (0.70) AURKAKIF11IDH2THRBLMNA
SCHEMBL6231959 0.77 RAPGEF4 (0.49) AURKANFKB1GRM4RAPGEF4
SCHEMBL30754777 0.77 LMNA (0.65) AURKAKIF11IDH2THRBLMNA
SCHEMBL31501743 0.77 AURKA (0.72) AURKAKIF11IDH2THRBLMNA
SCHEMBL6663767 0.77 AURKA (0.72) AURKAKIF11IDH2THRBLMNA
SCHEMBL4238979 0.76 AURKA (0.67) AURKAKIF11IDH2THRBLMNA
SCHEMBL6240725 0.76 TDO2 (0.51) CYP3A4GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed