SCHEMBL6254589

SCHEMBL6254589

O=C(O)c1cccc(-c2ccc(C(=O)O)cc2Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.59
RXRB P28702 1/20 0.59
KMO O15229 1/20 0.56
TSHR P16473 1/20 0.55
SRD5A2 P31213 1/20 0.53
FOLH1 Q04609 1/20 0.51
TNKS2 Q9H2K2 1/20 0.51
ADH5 P11766 1/20 0.49
AKR1C3 P42330 2/20 0.49
AKR1C2 P52895 2/20 0.49
DDT P30046 1/20 0.49
HSD17B1 P14061 1/20 0.49
HSD17B2 P37059 1/20 0.49
PTGER1 P34995 1/20 0.48
KEAP1 Q14145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442436 0.90 SRD5A2 (0.62) RXRARXRBKMOSRD5A2PTGER1
SCHEMBL2044221 0.89 SRD5A2 (0.60) RXRARXRBKMOTSHRSRD5A2
SCHEMBL25598474 0.87 CNR2 (0.55) RXRARXRBTSHRSRD5A2TNKS2
SCHEMBL3208003 0.86 KMO (0.62) RXRARXRBKMOSRD5A2HSD17B1
SCHEMBL2371293 0.86 KMO (0.61) RXRARXRBKMOFOLH1PTGER1
SCHEMBL6253145 0.83 SRD5A2 (0.72) RXRARXRBTSHRSRD5A2FOLH1
SCHEMBL23380737 0.83 RXRA (0.64) RXRARXRBTSHRSRD5A2TNKS2
SCHEMBL2769863 0.82 TSHR (0.71) RXRARXRBTSHRSRD5A2TNKS2
Hydrochloric Acid SCHEMBL9812960 0.81 SRD5A2 (0.70) RXRARXRBTSHRSRD5A2FOLH1
SCHEMBL5841701 0.81 RXRA (0.57) RXRARXRBKMOTSHRFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569954-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-09-07 EP disclosed
WO-2004052921-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-06-24 WO disclosed