SCHEMBL6255595

SCHEMBL6255595

N#CC1(NC(=O)[CH]Cc2c(F)ccc(C(N)=O)c2F)CCOCC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.35
ANO1 Q5XXA6 5/20 0.34
CNR1 P21554 5/20 0.33
JAK2 O60674 2/20 0.32
JAK1 P23458 2/20 0.32
CTSC P53634 1/20 0.31
STAT6 P42226 1/20 0.31
OPRL1 P41146 1/20 0.30
AR P10275 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6252183 0.88 JAK2 (0.35) JAK2JAK1CTSC
SCHEMBL2924445 0.70 DGAT1 (0.36) JAK2JAK1
SCHEMBL6252505 0.67
SCHEMBL6250638 0.67 CNR1 (0.39) CNR2ANO1CNR1CTSC
SCHEMBL4246964 0.67 CTSL (0.37) CTSC
SCHEMBL4239023 0.67 CTSL (0.34) CTSC
SCHEMBL5361109 0.66 CTSS (0.35) CNR2ANO1CNR1CTSC
SCHEMBL6194995 0.66 DGAT1 (0.40)
SCHEMBL5361057 0.66 CTSS (0.35) CNR1CTSC
SCHEMBL4247124 0.65 CTSL (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569954-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-09-07 EP disclosed
WO-2004052921-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-06-24 WO disclosed