SCHEMBL6257693

SCHEMBL6257693

CCCNc1nc(NN)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.75

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.71
ADORA2B P29275 1/20 0.71
PGK1 P00558 4/20 0.66
PGK2 P07205 4/20 0.66
SLC29A1 Q99808 1/20 0.61
ADORA3 P0DMS8 3/20 0.60
ADORA1 P30542 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5388703 0.92 ADORA2B (0.60) ADORA2AADORA2BPGK1PGK2SLC29A1
SCHEMBL5389218 0.92 ADORA2A (0.74) ADORA2AADORA2BPGK1PGK2ADORA3
SCHEMBL7083928 0.92 ADORA2A (0.74) ADORA2AADORA2BPGK1PGK2ADORA3
SCHEMBL4806899 0.88 PGK1 (0.85) ADORA2BPGK1PGK2SLC29A1ADORA3
SCHEMBL5393072 0.88 ADORA3 (0.77) ADORA2AADORA2BADORA3ADORA1
SCHEMBL5389657 0.88 ADORA3 (0.77) ADORA2AADORA2BADORA3ADORA1
SCHEMBL6262523 0.86 ADORA1 (0.71) ADORA2AADORA2BPGK1PGK2ADORA3
SCHEMBL5386790 0.86 ADORA1 (0.71) ADORA2AADORA2BPGK1PGK2ADORA3
SCHEMBL6262513 0.86 ADORA1 (0.71) ADORA2AADORA2BPGK1PGK2ADORA3
SCHEMBL6262904 0.85 ADORA2A (0.70) ADORA2AADORA2BPGK1PGK2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414837-B1 ADENOSINE A3 RECEPTOR AGONISTS CV THERAPEUTICS INC (US) 2005-10-19 EP disclosed
EP-1414837-A1 ADENOSINE A3 RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2004-05-06 EP disclosed
WO-2003014137-A1 ADENOSINE A3 RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2003-02-20 WO disclosed