SCHEMBL626133

SCHEMBL626133

CCNC(=O)N1CCC(NCc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.47
PIK3CD O00329 3/20 0.38
PIK3CB P42338 2/20 0.37
PIK3CG P48736 1/20 0.37
RIPK1 Q13546 4/20 0.36
MAP3K12 Q12852 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624920 0.87 PIK3CA (0.46) PIK3CAPIK3CDRIPK1CDK2
SCHEMBL626581 0.84 FYN (0.47) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL625652 0.84 PIK3CA (0.49) PIK3CAPIK3CDPIK3CBMAP3K12
SCHEMBL626134 0.84 PIK3CA (0.50) PIK3CAPIK3CDPIK3CBPIK3CGRIPK1
SCHEMBL625280 0.83 PIK3CA (0.49) PIK3CAMAP3K12
SCHEMBL625862 0.81 PIK3CA (0.47) PIK3CAPIK3CDPIK3CBPIK3CGMAP3K12
SCHEMBL624427 0.76 PIK3CA (0.50) PIK3CAMAP3K12
SCHEMBL627329 0.75 PIK3CA (0.49) PIK3CA
SCHEMBL627327 0.75 PIK3CA (0.49) PIK3CA
SCHEMBL626006 0.73 PIK3CA (0.46) PIK3CAPIK3CDPIK3CBPIK3CGRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed