SCHEMBL624920

SCHEMBL624920

CC(C)(C)OC(=O)N1CCC(NCc2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.46
RIPK1 Q13546 5/20 0.45
EPHX2 P34913 1/20 0.40
SYK P43405 1/20 0.38
SFRP1 Q8N474 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
PIK3CD O00329 1/20 0.37
GPR119 Q8TDV5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626133 0.87 PIK3CA (0.47) PIK3CARIPK1CDK2PIK3CD
SCHEMBL625127 0.86 PIK3CA (0.48) PIK3CARIPK1SYKCCNA2CDK2
SCHEMBL624984 0.84 PIK3CA (0.48) PIK3CARIPK1
SCHEMBL624921 0.82 PIK3CA (0.49) PIK3CARIPK1GPR119
SCHEMBL625280 0.82 PIK3CA (0.49) PIK3CA
SCHEMBL625652 0.82 PIK3CA (0.49) PIK3CAPIK3CD
SCHEMBL625862 0.80 PIK3CA (0.47) PIK3CAPIK3CD
SCHEMBL625421 0.80 PIK3CA (0.52) PIK3CARIPK1GPR119
SCHEMBL626544 0.80 ACKR3 (0.55) PIK3CARIPK1
SCHEMBL622971 0.79 ALDH1A1 (0.41) CCNA2CDK2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed