SCHEMBL625652

SCHEMBL625652

Nc1ncc(-c2cnc3sc(CNC4CCNCC4)nn23)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.49
MAP3K12 Q12852 4/20 0.38
FYN P06241 3/20 0.36
MAP4K3 Q8IVH8 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625280 0.86 PIK3CA (0.49) PIK3CAMAP3K12
SCHEMBL625862 0.86 PIK3CA (0.47) PIK3CAMAP3K12FYNPIK3CDPIK3CB
SCHEMBL626133 0.84 PIK3CA (0.47) PIK3CAMAP3K12PIK3CDPIK3CB
SCHEMBL625235 0.84 FYN (0.52) PIK3CAFYN
SCHEMBL624920 0.82 PIK3CA (0.46) PIK3CAPIK3CD
SCHEMBL626701 0.81 MKNK1 (0.52) PIK3CAFYN
SCHEMBL625653 0.78 PIK3CA (0.54) PIK3CAMAP3K12
SCHEMBL626700 0.78 PIK3CA (0.52) PIK3CAMAP3K12
SCHEMBL625674 0.76 PIK3CA (0.50) PIK3CAMAP3K12FYN
SCHEMBL624388 0.75 PIK3CA (0.55) PIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed