SCHEMBL6259489

SCHEMBL6259489

FC(F)(F)c1nc([AsH]C2CC2)c2ncn(-c3cccc(OCc4ccccc4)c3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
GRM5 P41594 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
FAAH O00519 1/20 0.34
MGLL Q99685 1/20 0.34
XDH P47989 1/20 0.34
MCHR1 Q99705 1/20 0.34
NR1H4 Q96RI1 2/20 0.34
ALOX5 P09917 1/20 0.34
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
TSHR P16473 2/20 0.33
TTK P33981 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6252841 0.91 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL3137716 0.82 YTHDC1 (0.42) PDE4APDE4BPDE4CPDE4DJAK2
SCHEMBL3136332 0.79 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DGRM5
SCHEMBL6236030 0.79 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL6257278 0.78 YTHDC1 (0.40) PDE4DXDHALDH1A1HPGD
SCHEMBL27611797 0.76 CYP2D6 (0.48) PDE4APDE4BPDE4CPDE4DGRM5
SCHEMBL4543346 0.75 XDH (0.40) PDE4APDE4BPDE4CPDE4DGRM5
SCHEMBL6258341 0.74 ALDH1A1 (0.34) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL6253561 0.73 SCN9A (0.40) XDH
SCHEMBL3130876 0.72 TLR7 (0.43) PDE4APDE4BPDE4CPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1529049-A2 DERIVATIVES OF 2-TRIFLUORMETHYL-6-AMINOPURINE AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceutical Corporation (US) 2005-05-11 EP disclosed
WO-2004014913-A2 DERIVATIVES OF 2-TRIFLUORMETHYL-6-AMINOPURINE AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-02-19 WO disclosed