SCHEMBL626135

SCHEMBL626135

CCNC(=O)N1CCC(N(C)c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.45
MAP3K12 Q12852 14/20 0.41
PIK3CD O00329 2/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
DLK1 P80370 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626134 0.85 PIK3CA (0.50) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL624922 0.85 PIK3CA (0.42) PIK3CAMAP3K12
SCHEMBL626582 0.84 PIK3CA (0.42) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL625654 0.83 MAP3K12 (0.47) PIK3CAMAP3K12DLK1
SCHEMBL626637 0.83 MAP3K12 (0.47) PIK3CAMAP3K12DLK1
SCHEMBL625051 0.82 MAP3K12 (0.46) PIK3CAMAP3K12DLK1
SCHEMBL625282 0.81 MAP3K12 (0.45) PIK3CAMAP3K12DLK1
SCHEMBL625864 0.80 MAP3K12 (0.44) PIK3CAMAP3K12DLK1
SCHEMBL627783 0.80 MAP3K12 (0.46) PIK3CAMAP3K12DLK1
SCHEMBL627328 0.75 PIK3CA (0.44) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed