SCHEMBL627328

SCHEMBL627328

CCNC(=O)NC1CCC(Nc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.44
MAP3K12 Q12852 12/20 0.41
PIK3CD O00329 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
DLK1 P80370 1/20 0.38
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38
CYP3A4 P08684 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627397 0.89 PIK3CA (0.49) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL626892 0.85 PIK3CA (0.42) PIK3CAMAP3K12DLK1CYP3A4MAP4K1
SCHEMBL627440 0.85 FYN (0.45) PIK3CAMAP3K12DLK1
SCHEMBL627329 0.85 PIK3CA (0.49) PIK3CA
SCHEMBL627327 0.85 PIK3CA (0.49) PIK3CA
SCHEMBL624428 0.83 MAP3K12 (0.47) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL625301 0.83 MAP3K12 (0.44) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL625636 0.82 MAP3K12 (0.44) PIK3CAMAP3K12DLK1MAP4K1
SCHEMBL626299 0.82 PIK3CA (0.47) PIK3CAMAP3K12PIK3CDPIK3CBPIK3CG
SCHEMBL626007 0.82 MAPT (0.51) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed