SCHEMBL624922

SCHEMBL624922

CN(c1nn2cc(-c3cnc(N)c(C(F)(F)F)c3)nc2s1)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.42
MAP3K12 Q12852 8/20 0.41
RIPK1 Q13546 2/20 0.40
GPR119 Q8TDV5 7/20 0.40
MAP4K1 Q92918 1/20 0.39
USP30 Q70CQ3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624921 0.85 PIK3CA (0.49) PIK3CAMAP3K12RIPK1GPR119
SCHEMBL626135 0.85 PIK3CA (0.45) PIK3CAMAP3K12
SCHEMBL625128 0.85 CCNA2 (0.46) PIK3CAMAP3K12RIPK1GPR119MAP4K1
SCHEMBL626637 0.84 MAP3K12 (0.47) PIK3CAMAP3K12
SCHEMBL625422 0.83 PIK3CA (0.42) PIK3CAMAP3K12
SCHEMBL625051 0.83 MAP3K12 (0.46) PIK3CAMAP3K12MAP4K1
SCHEMBL624985 0.83 KDM4E (0.40) PIK3CAMAP3K12GPR119MAP4K1
SCHEMBL627783 0.82 MAP3K12 (0.46) PIK3CAMAP3K12
SCHEMBL625654 0.82 MAP3K12 (0.47) PIK3CAMAP3K12
SCHEMBL625282 0.81 MAP3K12 (0.45) PIK3CAMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed