SCHEMBL626212

SCHEMBL626212

CC(C)(C)OC(=O)NC(c1nn2c(I)cnc2s1)C1CCCNC1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.33
CDK2 P24941 1/20 0.31
AKT1 P31749 1/20 0.31
IRAK4 Q9NWZ3 6/20 0.30
CHEK1 O14757 2/20 0.30
BTK Q06187 2/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626888 0.89 AAK1 (0.34) AAK1AKT1JAK2JAK1
SCHEMBL17764699 0.70 AAK1 (0.37) AAK1CDK2AKT1BTK
SCHEMBL625036 0.69 PIM1 (0.49)
SCHEMBL625189 0.69 PIK3CA (0.46)
SCHEMBL17764670 0.69 AXL (0.42) AAK1CDK2IRAK4CHEK1
SCHEMBL627106 0.69 FYN (0.44) BTKJAK2JAK1
SCHEMBL626398 0.69 FYN (0.44) BTKJAK2JAK1
SCHEMBL15719996 0.69 PDE2A (0.42)
SCHEMBL3955485 0.68 CPN1 (0.39) AAK1BTK
SCHEMBL627225 0.68 CKS1B (0.48) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed