SCHEMBL626299

SCHEMBL626299

CCNC(=O)NCCNc1nn2cc(-c3cnc(N)c(C(F)(F)F)c3)nc2s1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.47
PIK3CD O00329 2/20 0.42
PIK3CB P42338 2/20 0.42
PIK3CG P48736 2/20 0.42
CYP3A4 P08684 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
MAP3K12 Q12852 7/20 0.40
F2RL3 Q96RI0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625400 0.86 PIK3CA (0.43) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626145 0.84 F2RL3 (0.43) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626269 0.84 F2RL3 (0.44) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL624442 0.84 PIK3CA (0.44) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626298 0.84 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL627328 0.82 PIK3CA (0.44) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL12474086 0.82 PIK3CA (0.47) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626774 0.81 PIK3CA (0.42) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626625 0.81 PIK3CA (0.43) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4
SCHEMBL626582 0.81 PIK3CA (0.42) PIK3CAPIK3CDPIK3CBPIK3CGCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed