SCHEMBL6266372

SCHEMBL6266372

CCOC(=O)C1=CCN(C(=O)O)C=CC1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
ALDH1A1 P00352 7/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HSP90AA1 P07900 1/20 0.35
CACNA1B Q00975 1/20 0.35
APBA1 Q02410 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GAA P10253 3/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
MAPT P10636 3/20 0.33
LMNA P02545 2/20 0.33
ADORA2B P29275 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPC5 Q9UL62 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28039152 0.66 KDM4E (0.44) TSHRALDH1A1KDM4EHPGDHTT
SCHEMBL9626894 0.65 TSHR (0.48) TSHRALDH1A1KDM4EHPGDHTT
SCHEMBL31196992 0.65 TSHR (0.48) TSHRALDH1A1KDM4EHPGDTDP1
SCHEMBL6180556 0.65 ALDH1A1 (0.37) TSHRALDH1A1KDM4EHPGDTDP1
SCHEMBL15764230 0.65 KDM4E (0.40) TSHRALDH1A1KDM4EHPGDHTT
SCHEMBL27672566 0.63 ALDH1A1 (0.36) TSHRALDH1A1KDM4EHTTTDP1
SCHEMBL819891 0.62 TSHR (0.45) TSHRALDH1A1KDM4EHPGDTDP1
SCHEMBL15157001 0.62 RAB9A (0.33) TSHRALDH1A1KDM4EHPGDHTT
SCHEMBL5338308 0.62 KMT2A (0.42) TSHRALDH1A1KDM4EHPGDBAZ2B
SCHEMBL11438318 0.62 TSHR (0.38) TSHRALDH1A1KDM4EHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558577-A2 SUBSTITUTED 4-PHENYL-PIPERIDIN-AMIDES AS TACHYKININ ANTAGONISTS AND SEROTONIN REPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-08-03 EP disclosed
WO-2004005256-A2 SUBSTITUTED 4-PHENYL-PIPERIDIN-AMIDES AS TACHYKININ ANTAGONISTS AND SEROTONIN REPTAKE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-01-15 WO disclosed