SCHEMBL626703

SCHEMBL626703

CN1CCN(c2ncc(-c3cnc4sc(NC5CCN(S(C)(=O)=O)CC5)nn34)cc2C(F)(F)F)CC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.53
FYN P06241 11/20 0.44
CCNE1 P24864 5/20 0.42
CDK2 P24941 5/20 0.42
CCND1 P24385 2/20 0.42
CDK6 Q00534 2/20 0.42
CDK1 P06493 1/20 0.42
CDK4 P11802 1/20 0.42
CCNB1 P14635 1/20 0.42
CCND3 P30281 1/20 0.42
HASPIN Q8TF76 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624393 0.91 FYN (0.46) PIK3CAFYNCCNE1CDK2CCND1
SCHEMBL625860 0.89 GPR119 (0.47) PIK3CAFYNHASPIN
SCHEMBL626206 0.86 PIK3CA (0.53) PIK3CAFYNHASPIN
SCHEMBL626704 0.85 CCNE1 (0.43) PIK3CACCNE1CDK2CCND1CDK6
SCHEMBL626164 0.81 FYN (0.51) FYNCCNE1CDK2CCND1CDK6
SCHEMBL625753 0.77 PIK3CA (0.49) PIK3CAFYNHASPIN
SCHEMBL624394 0.77 CCNE1 (0.41) CCNE1CDK2CCND1CDK6CDK1
SCHEMBL626171 0.77 FYN (0.54) FYNHASPIN
SCHEMBL625861 0.75 GPR119 (0.46) CCNE1CDK2CCND1CDK6CDK1
SCHEMBL624430 0.74 FYN (0.72) PIK3CAFYNHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed