SCHEMBL626704

SCHEMBL626704

CN1CCN(c2ncc(-c3cn4nc(NC5CCN(S(C)(=O)=O)CC5)sc4n3)cc2C(F)(F)F)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 17/20 0.43
CDK2 P24941 17/20 0.43
CDK1 P06493 10/20 0.43
CCNB1 P14635 10/20 0.43
CCND1 P24385 10/20 0.43
CDK6 Q00534 10/20 0.43
CDK4 P11802 8/20 0.43
CCND3 P30281 8/20 0.43
PIK3CA P42336 1/20 0.39
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
IDO1 P14902 1/20 0.37
CCNT1 O60563 2/20 0.36
CDK7 P50613 2/20 0.36
CDK9 P50750 2/20 0.36
CCNH P51946 2/20 0.36
MNAT1 P51948 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624394 0.92 CCNE1 (0.41) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL625861 0.89 GPR119 (0.46) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL626207 0.87 MAP3K12 (0.46) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL626703 0.85 PIK3CA (0.53) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL626165 0.81 IDO1 (0.47) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL625754 0.78 MAP3K12 (0.40) PIK3CA
SCHEMBL626172 0.77 DYRK1A (0.38) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL624393 0.77 FYN (0.46) CCNE1CDK2CDK1CCNB1CCND1
SCHEMBL624428 0.75 MAP3K12 (0.47) PIK3CA
SCHEMBL625860 0.75 GPR119 (0.47) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed