SCHEMBL625861

SCHEMBL625861

CC(C)(C)OC(=O)N1CCN(c2ncc(-c3cn4nc(NC5CCN(S(C)(=O)=O)CC5)sc4n3)cc2C(F)(F)F)CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.46
SYK P43405 1/20 0.39
CDK2 P24941 9/20 0.38
CCNE1 P24864 8/20 0.38
CCND1 P24385 5/20 0.38
CDK6 Q00534 5/20 0.38
CDK1 P06493 5/20 0.38
CCNB1 P14635 5/20 0.38
CDK4 P11802 4/20 0.38
CCND3 P30281 4/20 0.38
IDH1 O75874 1/20 0.37
IDH2 P48735 1/20 0.37
SFRP1 Q8N474 1/20 0.36
CCNA2 P20248 1/20 0.36
ALK Q9UM73 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626704 0.89 CCNE1 (0.43) CDK2CCNE1CCND1CDK6CDK1
SCHEMBL624394 0.87 CCNE1 (0.41) CDK2CCNE1CCND1CDK6CDK1
SCHEMBL625860 0.86 GPR119 (0.47) GPR119SYK
SCHEMBL625128 0.85 CCNA2 (0.46) GPR119SYKCDK2IDH1IDH2
SCHEMBL625456 0.83 MAP3K12 (0.41) GPR119SYKCDK2CCNE1CCND1
SCHEMBL626207 0.83 MAP3K12 (0.46) CDK2CCNE1CCND1CDK6CDK1
SCHEMBL625408 0.77 MAP4K1 (0.39) SYKCDK2CCNA2
SCHEMBL626165 0.77 IDO1 (0.47) CDK2CCNE1CCND1CDK6CDK1
SCHEMBL2121138 0.76 PIK3CA (0.56) ALK
SCHEMBL626703 0.75 PIK3CA (0.53) CDK2CCNE1CCND1CDK6CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed