SCHEMBL626892

SCHEMBL626892

CC(C)(C)OC(=O)NC1CCC(Nc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.42
MAP3K12 Q12852 15/20 0.41
DLK1 P80370 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627397 0.89 PIK3CA (0.49) PIK3CAMAP3K12DLK1CYP3A4
SCHEMBL625128 0.88 CCNA2 (0.46) PIK3CAMAP3K12MAP4K1
SCHEMBL625132 0.86 CKS1B (0.42) PIK3CAMAP3K12
SCHEMBL627328 0.85 PIK3CA (0.44) PIK3CAMAP3K12DLK1CYP3A4MAP4K1
SCHEMBL627440 0.85 FYN (0.45) PIK3CAMAP3K12DLK1
SCHEMBL626893 0.85 PIK3CA (0.49) PIK3CA
SCHEMBL626891 0.85 PIK3CA (0.49) PIK3CA
SCHEMBL624991 0.83 SYK (0.45) PIK3CAMAP3K12
SCHEMBL624428 0.83 MAP3K12 (0.47) PIK3CAMAP3K12DLK1CYP3A4
SCHEMBL625301 0.83 MAP3K12 (0.44) PIK3CAMAP3K12DLK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed