SCHEMBL624428

SCHEMBL624428

CC(=O)N1CCC(Nc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 14/20 0.47
PIK3CA P42336 5/20 0.46
SYK P43405 1/20 0.41
CYP3A4 P08684 1/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41
PIK3CG P48736 1/20 0.41
DLK1 P80370 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625128 0.89 CCNA2 (0.46) MAP3K12PIK3CASYK
SCHEMBL627397 0.89 PIK3CA (0.49) MAP3K12PIK3CACYP3A4PIK3CDPIK3CB
SCHEMBL626207 0.87 MAP3K12 (0.46) MAP3K12PIK3CA
SCHEMBL627440 0.87 FYN (0.45) MAP3K12PIK3CADLK1
SCHEMBL625301 0.86 MAP3K12 (0.44) MAP3K12PIK3CACYP3A4PIK3CDPIK3CB
SCHEMBL625636 0.85 MAP3K12 (0.44) MAP3K12PIK3CADLK1
SCHEMBL625236 0.85 MAP3K12 (0.45) MAP3K12PIK3CADLK1
SCHEMBL624427 0.84 PIK3CA (0.50) MAP3K12PIK3CA
SCHEMBL625754 0.84 MAP3K12 (0.40) MAP3K12PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL627328 0.83 PIK3CA (0.44) MAP3K12PIK3CACYP3A4PIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed