SCHEMBL626985

SCHEMBL626985

c1cc(-c2cn3nc(N4CCOCC4)sc3n2)c2cn[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.53
PIK3R1 P27986 8/20 0.53
PIK3CD O00329 5/20 0.51
PIK3CB P42338 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
MTOR P42345 2/20 0.46
PIK3CG P48736 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626984 0.80 PIK3CA (0.48) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL893058 0.73 PIK3CA (0.72) PIK3CAPIK3R1PIK3CDPIK3CBHDAC6
SCHEMBL10100419 0.72 ROCK2 (0.71) PIK3CAPIK3R1PIK3CDPIK3CBHDAC6
SCHEMBL625392 0.72 F2RL3 (0.42) MTOR
SCHEMBL1309601 0.71 PIK3CA (0.60) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL625797 0.71 PIK3CA (0.53) PIK3CAPIK3R1PIK3CDPIK3CBHDAC6
SCHEMBL1309278 0.71 PIK3CA (0.77) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL18193255 0.71 PIK3CA (0.76) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL20458892 0.71 PIK3CA (0.61) PIK3CAPIK3R1PIK3CDPIK3CBHDAC6
SCHEMBL893372 0.71 PIK3CA (0.69) PIK3CAPIK3R1PIK3CDPIK3CBHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed