SCHEMBL626984

SCHEMBL626984

c1cc(-c2cnc3sc(N4CCOCC4)nn23)c2cn[nH]c2c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 16/20 0.48
PIK3CB P42338 2/20 0.48
PIK3CG P48736 2/20 0.47
PIK3CD O00329 2/20 0.47
HASPIN Q8TF76 3/20 0.46
MTOR P42345 2/20 0.45
PIK3R1 P27986 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626985 0.80 PIK3CA (0.53) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL625391 0.76 HASPIN (0.52) HASPIN
SCHEMBL625796 0.73 PIK3CA (0.47) PIK3CAPIK3CD
SCHEMBL18193255 0.69 PIK3CA (0.76) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL1309278 0.69 PIK3CA (0.77) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL4075802 0.69 AR (0.55) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL1310548 0.69 ATR (0.58) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL624034 0.68 LMNA (0.48)
SCHEMBL10100419 0.67 ROCK2 (0.71) PIK3CAPIK3CBPIK3CGPIK3CDMTOR
SCHEMBL19142657 0.67 PIK3CA (0.65) PIK3CAPIK3CBPIK3CGPIK3CDMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed