SCHEMBL6270127

SCHEMBL6270127

O=C(/C=C\c1cccnc1)NCCCCN1CCC(c2cccc3ccccc23)CC1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 18/20 0.59
DRD2 P14416 1/20 0.55
DRD3 P35462 1/20 0.55
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
NAMPT P43490 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL88313 0.86 CCR2 (0.81) CCR2DRD2DRD3
SCHEMBL88314 0.86 CCR2 (0.81) CCR2DRD2DRD3
SCHEMBL83120 0.86 DRD3 (0.62) CCR2DRD2DRD3CYP3A4CYP2C9
SCHEMBL3079779 0.86 DRD3 (0.62) CCR2DRD2DRD3CYP3A4CYP2C9
SCHEMBL3090708 0.84 DRD2 (0.71) DRD2DRD3
SCHEMBL82403 0.84 DRD2 (0.71) DRD2DRD3
SCHEMBL6264932 0.84 DRD2 (0.51) CCR2DRD2DRD3CYP3A4CYP2C9
SCHEMBL6264935 0.84 DRD2 (0.51) CCR2DRD2DRD3CYP3A4CYP2C9
SCHEMBL6267972 0.82 DRD3 (0.57) CCR2DRD2DRD3CYP3A4CYP2C9
SCHEMBL6267971 0.82 DRD3 (0.57) CCR2DRD2DRD3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1079832-B1 USE OF VITAMIN PP COMPOUNDS KLINGE CO CHEM PHARM FAB (DE) 2005-11-30 EP claimed