SCHEMBL6270519

SCHEMBL6270519

Fc1cccc(F)c1-c1cnnc(-c2ccc(-c3ccc(OC(F)(F)F)cc3)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 11/20 0.39
TYK2 P29597 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SCN1A P35498 1/20 0.36
SCN2A Q99250 1/20 0.36
CYP1A2 P05177 1/20 0.35
CHRNA7 P36544 3/20 0.35
ACP1 P24666 1/20 0.35
CASP3 P42574 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6762808 0.82 ALOX5AP (0.39) SCN5ATYK2ADORA3KDM4ENPC1
SCHEMBL6271045 0.77 ADORA2A (0.45) NPC1ALDH1A1GAAMAPTRAB9A
SCHEMBL6266948 0.76 ALOX5AP (0.39) SCN5ATYK2KDM4ENPC1ALDH1A1
SCHEMBL4391246 0.76 TYK2 (0.45) SCN5ATYK2KDM4ENPC1ALDH1A1
SCHEMBL2645021 0.73 DYRK1A (0.48) KDM4EALDH1A1MAPTRAB9ACHRNA7
SCHEMBL2645408 0.67 ATR (0.45) CYP1A2ALOX5APFEN1
SCHEMBL4613467 0.66 TDP2 (0.46) SCN5ATYK2NPC1ALDH1A1RAB9A
SCHEMBL3664986 0.65 CLK4 (0.57) SCN5AKDM4ENPC1ALDH1A1GAA
SCHEMBL29628993 0.64 SCN5A (0.54) SCN5AALDH1A1SCN1ASCN2A
SCHEMBL7696321 0.64 NISCH (0.43) SCN5ATYK2KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175410-B1 PESTICIDAL TRIAZINE DERIVATIVES NOVARTIS AG (CH) 2005-12-07 EP disclosed
US-6723720-B2 PHENYL-SUBSTITUTED 1,2,4-TRIAZINES, ESPECIALLY FOR CONTROLLING FLEAS NOVARTIS ANIMAL HEALTH US, INC. 2004-04-20 US disclosed
US-20030036544-A1 Pesticidal triazine-derivatives NOVARTIS ANIMAL HEALTH US, INC. 2003-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030036544-A1 Pesticidal triazine-derivatives DDT, CYCS, TUBA3C SCN5A 807/4885TYK2 3815/4885ADORA3 2377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.