SCHEMBL6270691

SCHEMBL6270691

O=C(NC(=O)N1CCN(C(=O)c2ccccc2)C(C(=O)NC(c2ccccc2)c2ccccc2)C1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
CACNA2D1 P54289 2/20 0.43
CACNA1B Q00975 2/20 0.43
CACNB1 Q02641 2/20 0.43
CACNA1C Q13936 1/20 0.43
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
XIAP P98170 4/20 0.41
BIRC3 Q13489 2/20 0.41
BIRC2 Q13490 2/20 0.41
LMNA P02545 2/20 0.40
HTT P42858 1/20 0.40
MAOB P27338 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CFD P00746 1/20 0.39
HPGDS O60760 1/20 0.39
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038814 0.84 AGTR2 (0.44) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4041221 0.81 ALDH1A1 (0.49) GAAALDH1A1LMNA
SCHEMBL4034993 0.80 CACNA2D1 (0.48) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4035592 0.75 ALDH1A1 (0.53) GAAALDH1A1SMN1; SMN2XIAPBIRC3
SCHEMBL4032376 0.73 ALDH1A1 (0.53) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4037091 0.71 ENPP2 (0.46) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4032714 0.70 HTR1A (0.44) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL13197309 0.68 XIAP (0.57) XIAPBIRC3BIRC2
SCHEMBL17512449 0.67 CACNA2D1 (0.81) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4032488 0.67 POLB (0.46) ALDH1A1SMN1; SMN2MEN1KMT2ACFD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2005-11-09 EP disclosed
WO-2004071390-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-08-26 WO disclosed