SCHEMBL627267

SCHEMBL627267

CC(C)(C)OC(=O)N1CCC2(CC1)CN(c1nn3cc(I)nc3s1)C2

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.41
ACACB O00763 5/20 0.41
SCD5 Q86SK9 1/20 0.40
RET P07949 8/20 0.39
SPR P35270 3/20 0.38
USP2 O75604 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627422 0.93 RET (0.42) CYP11B2ACACBSCD5RETUSP2
SCHEMBL628407 0.93 CYP11B2 (0.44) CYP11B2ACACBSCD5RETCYP3A4
SCHEMBL627265 0.87 CKS1B (0.41)
SCHEMBL625492 0.81 NAMPT (0.39) ACACB
SCHEMBL627207 0.80 OPRM1 (0.39) SPR
SCHEMBL627266 0.80 CYP11B2 (0.41) CYP11B2ACACBSCD5RETSPR
SCHEMBL627513 0.77 OPRM1 (0.37)
SCHEMBL627020 0.77 RET (0.40) RETHDAC1HDAC2
SCHEMBL627341 0.76 NAMPT (0.47)
SCHEMBL627421 0.75 RET (0.44) CYP11B2ACACBRETUSP2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed