SCHEMBL628407

SCHEMBL628407

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3cc(I)nc3s1)CC2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.44
RET P07949 2/20 0.39
ACACB O00763 5/20 0.38
CYP3A4 P08684 1/20 0.37
GPR119 Q8TDV5 4/20 0.37
SCD5 Q86SK9 1/20 0.37
KIF18A Q8NI77 1/20 0.37
HIF1A Q16665 1/20 0.36
NAMPT P43490 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627267 0.93 CYP11B2 (0.41) CYP11B2RETACACBCYP3A4SCD5
SCHEMBL627265 0.90 CKS1B (0.41) GPR119
SCHEMBL627422 0.90 RET (0.42) CYP11B2RETACACBCYP3A4SCD5
SCHEMBL625492 0.81 NAMPT (0.39) ACACBGPR119NAMPT
SCHEMBL627207 0.81 OPRM1 (0.39) GPR119
SCHEMBL628406 0.79 CYP11B2 (0.44) CYP11B2RETACACBCYP3A4GPR119
SCHEMBL627513 0.78 OPRM1 (0.37) GPR119
SCHEMBL627341 0.77 NAMPT (0.47) GPR119NAMPTJAK2JAK1
SCHEMBL625512 0.76 THRB (0.44) CYP11B2SCD5
SCHEMBL627226 0.75 CKS1B (0.46) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed