SCHEMBL627309

SCHEMBL627309

CC(C)(C)OC(=O)N1CC2CN(c3nn4cc(-c5cnc(N)c(C(F)(F)F)c5)nc4s3)CC2C1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 16/20 0.46
PIK3CA P42336 2/20 0.41
DLK1 P80370 1/20 0.38
USP30 Q70CQ3 1/20 0.38
MAP4K1 Q92918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625422 0.89 PIK3CA (0.42) MAP3K12PIK3CA
SCHEMBL627308 0.87 PIK3CA (0.49) MAP3K12PIK3CAUSP30
SCHEMBL626246 0.86 MAP3K12 (0.40) MAP3K12PIK3CADLK1
SCHEMBL627432 0.85 RET (0.40) MAP3K12PIK3CADLK1MAP4K1
SCHEMBL627020 0.85 RET (0.40) MAP3K12PIK3CA
SCHEMBL626620 0.84 MAP3K12 (0.52) MAP3K12PIK3CADLK1
SCHEMBL626123 0.82 RET (0.43) MAP3K12PIK3CA
SCHEMBL624991 0.81 SYK (0.45) MAP3K12PIK3CA
SCHEMBL625132 0.81 CKS1B (0.42) MAP3K12PIK3CA
SCHEMBL624922 0.80 PIK3CA (0.42) MAP3K12PIK3CAUSP30MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed