SCHEMBL627340

SCHEMBL627340

CC(C)(C)OC(=O)N1CCC2(CC1)CC(CNc1nn3c(I)cnc3s1)C2

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.49
GPR119 Q8TDV5 6/20 0.43
ACKR3 P25106 2/20 0.41
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627066 0.88 KDM4E (0.46) GPR119ACKR3
SCHEMBL625491 0.86 NAMPT (0.41) NAMPTGPR119ACKR3CYP2C9
SCHEMBL627341 0.82 NAMPT (0.47) NAMPTGPR119ACKR3CYP2C9
SCHEMBL624453 0.80 PIM1 (0.51)
SCHEMBL627014 0.79 ACKR3 (0.63) GPR119ACKR3
SCHEMBL627262 0.77 CCNA2 (0.48) GPR119ACKR3
SCHEMBL628406 0.77 CYP11B2 (0.44) GPR119
SCHEMBL627266 0.76 CYP11B2 (0.41) GPR119
SCHEMBL627421 0.73 RET (0.44) CYP2C9
SCHEMBL622971 0.73 ALDH1A1 (0.41) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed