SCHEMBL6280822

SCHEMBL6280822

CC(C)c1ccc(/C=C(/C(N)=O)C(=O)N(c2cccc(C(F)(F)F)c2)c2ccc3[nH]ccc3c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.35
GLI1 P08151 1/20 0.34
GLI2 P10070 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ESR1 P03372 1/20 0.33
PTGS2 P35354 1/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 2/20 0.33
CCR2 P41597 1/20 0.31
RECQL P46063 1/20 0.30
EPHX1 P07099 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6280828 1.00 IDH1 (0.35) IDH1GLI1GLI2TRPV1ESR1
SCHEMBL6248753 0.88 EPHX1 (0.37) CCR2RECQLEPHX1LMNAMAPT
SCHEMBL6245831 0.78 MAPT (0.35) PTGS2LMNATP53MAPT
SCHEMBL6247880 0.76 RECQL (0.43) RECQLLMNAMAPT
SCHEMBL5142623 0.76 IDH1 (0.52) IDH1TRPV1ESR1LMNATP53
SCHEMBL5142626 0.76 IDH1 (0.52) IDH1TRPV1ESR1LMNATP53
SCHEMBL6246748 0.73 GRK2 (0.40) RECQLLMNAMAPT
SCHEMBL6246353 0.73 RORC (0.40) IDH1RECQL
SCHEMBL6246114 0.72 ALDH1A1 (0.48) LMNAMAPT
SCHEMBL6248097 0.71 PTGS1 (0.44) RECQLLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO disclosed