SCHEMBL6246353

SCHEMBL6246353

N#Cc1ccc(C=C(C(N)=O)C(=O)N(c2cccc(C(F)(F)F)c2)c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.40
RPS6KA3 P51812 1/20 0.38
JAK3 P52333 1/20 0.38
ELANE P08246 9/20 0.37
RXFP1 Q9HBX9 1/20 0.37
VNN1 O95497 1/20 0.37
RECQL P46063 1/20 0.37
CYP2C9 P11712 3/20 0.37
CYP3A4 P08684 2/20 0.36
ERBB2 P04626 1/20 0.36
IDH1 O75874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6247880 0.86 RECQL (0.43) RECQL
SCHEMBL6246748 0.83 GRK2 (0.40) RORCRXFP1VNN1RECQLCYP2C9
SCHEMBL6248753 0.83 EPHX1 (0.37) RECQL
SCHEMBL6246114 0.82 ALDH1A1 (0.48)
SCHEMBL6265380 0.80 LMNA (0.41)
SCHEMBL6248097 0.78 PTGS1 (0.44) RXFP1RECQLCYP3A4
SCHEMBL6246207 0.78 LMNA (0.34) RECQL
SCHEMBL6244821 0.77 NQO2 (0.46) RORCRXFP1CYP2C9CYP3A4
SCHEMBL6248564 0.76 MAPT (0.43) RORCRXFP1RECQL
SCHEMBL6247079 0.76 JAK2 (0.38) RORCRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037196-A2 SUBSTITUTED 2-ARYLMETHYLENE-N-ARYL-N'-ARYL-MALONAMIDES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS CYTOVIA, INC. (US) 2005-04-28 WO claimed