SCHEMBL6283903

SCHEMBL6283903

CC(C)Oc1cccc(-n2c(=S)[nH]c3ccccc3c2=O)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.63
PDE7B Q9NP56 1/20 0.63
HTT P42858 2/20 0.60
NPSR1 Q6W5P4 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
MAPT P10636 1/20 0.60
CYP2C9 P11712 1/20 0.60
ALOX12 P18054 1/20 0.60
CYP2C19 P33261 1/20 0.60
CA12 O43570 2/20 0.59
CA1 P00915 2/20 0.59
CA2 P00918 2/20 0.59
CA9 Q16790 2/20 0.59
RXFP1 Q9HBX9 2/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 4/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6276511 0.86 PDE7A (0.68) PDE7APDE7BHTTNPSR1ALOX12
SCHEMBL6278508 0.81 LOXL3 (0.65) HTTCYP1A2MAPTCYP2C9CYP2C19
SCHEMBL30103233 0.78 PDE7A (1.00) PDE7APDE7BHTTNPSR1MAPT
SCHEMBL844588 0.78 PDE7A (1.00) PDE7APDE7BHTTNPSR1MAPT
SCHEMBL6283951 0.78 PDE7A (0.71) PDE7APDE7BHTTNPSR1CA12
SCHEMBL6306891 0.78 PDE7A (0.71) PDE7APDE7BHTTNPSR1CA12
SCHEMBL6279687 0.78 PDE7A (0.66) PDE7APDE7BHTTNPSR1CA12
SCHEMBL6278489 0.76 KMT2A (0.75) PDE7APDE7BHTTNPSR1MAPT
SCHEMBL6280615 0.75 ALDH1A1 (0.65) PDE7APDE7BHTTNPSR1CYP1A2
SCHEMBL6281073 0.74 PDE7A (0.64) PDE7APDE7BHTTNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897213-B1 Heterocycles as cholecystokinin (CCK) ligands WARNER-LAMBERT COMPANY (US) 2005-05-24 US disclosed
US-5869665-A REACTING 2-HYDRAZINE PRECURSOR WITH HYDROGEN; CYCLIZATION WARNER-LAMBERT COMPANY (US) 1999-02-09 US disclosed
US-5756502-A APPETITE SUPPRESSANTS AND ANTISECRETORY AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-26 US disclosed
WO-1996020178-A1 NOVEL HETEROCYCLES AS CHOLECYSTOKININ (CCK) LIGANDS WARNER-LAMBERT COMPANY (US) 1996-07-04 WO disclosed