Anthranilamide

Anthranilamide

SCHEMBL6284801

COc1cccc2cc(C(=O)O)sc12.NC(=O)c1ccccc1N

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
KDM4E B2RXH2 4/20 0.42
HPGD P15428 3/20 0.42
HTT P42858 1/20 0.42
CHRNA7 P36544 3/20 0.41
HSD17B10 Q99714 3/20 0.41
CFTR P13569 1/20 0.41
BCL2L1 Q07817 1/20 0.40
HTR3A P46098 1/20 0.40
RCE1 Q9Y256 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
PARP1 P09874 1/20 0.39
IKBKB O14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6284804 0.90 CA2 (0.49) CA2ALDH1A1KMT2AADORA1KDM4E
SCHEMBL1850788 0.84 CA2 (0.53) CA2ALDH1A1KMT2AADORA1KDM4E
Anthranilamide SCHEMBL6288989 0.83 STING1 (0.49) ALDH1A1HSD17B10CFTRBCL2L1
SCHEMBL17858541 0.79 BCL2L1 (0.50) ALDH1A1KDM4EBCL2L1NPC1RAB9A
Anthranilamide SCHEMBL6280290 0.78 KMT2A (0.67) CA2ALDH1A1KMT2AADORA2AADORA2B
SCHEMBL15697569 0.77 BCL2L1 (0.46) CA2ALDH1A1KMT2AKDM4EHPGD
SCHEMBL3252698 0.76 BCL2L1 (0.53) CA2ALDH1A1KMT2AKDM4EHPGD
SCHEMBL3254246 0.75 GAA (0.57) ALDH1A1KMT2AHPGDHSD17B10NPC1
SCHEMBL2895989 0.75 ALDH1A1 (0.55) CA2ALDH1A1KMT2AADORA1KDM4E
SCHEMBL6284802 0.75 LMNA (0.51) CA2ALDH1A1ADORA1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2005508311-A 2005-03-31 JP claimed
EP-1416928-A2 N-MONOACYLATED DERIVATIVES OF O-PHENYLENEDIAMINES, THEIR SIX MEMBERED HETEROCYCLIC ANALOGUES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2004-05-12 EP claimed
WO-2003013484-A2 N-MONOACYLATED DERIVATIVES OF O-PHENYLENEDIAMINES, THEIR SIX MEMBERED HETEROCYCLIC ANALOGUES AND THEIR USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2003-02-20 WO claimed