SCHEMBL6285067

SCHEMBL6285067

COC(=O)[C@@H]1CCC[N+]1(C(=O)OC)C(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CPB1 P15086 1/20 0.44
FKBP1A P62942 4/20 0.43
TSHR P16473 3/20 0.42
ALDH1A1 P00352 5/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP2D6 P10635 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CASP1 P29466 1/20 0.39
GAA P10253 1/20 0.39
LMNA P02545 1/20 0.38
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806227 0.84 SMN1; SMN2 (0.45) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL2438026 0.79 CPB1 (0.41) CPB1FKBP1ATSHRALDH1A1CYP2C9
SCHEMBL696626 0.79 CYP3A4 (0.40) FKBP1ATSHRALDH1A1CYP2C9CYP2C19
SCHEMBL3295119 0.77 CYP2C19 (0.45) FKBP1ATSHRALDH1A1CYP2C9CYP2C19
SCHEMBL18281695 0.77 KMT2A (0.43) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL15665799 0.74 ALDH1A1 (0.44) FKBP1ATSHRALDH1A1CYP2C9CYP2C19
SCHEMBL15665561 0.74 ALDH1A1 (0.44) FKBP1ATSHRALDH1A1CYP2C9CYP2C19
SCHEMBL489617 0.73 SMN1; SMN2 (0.42) CPB1FKBP1ATSHRALDH1A1CYP3A4
SCHEMBL6810385 0.72 ALDH1A1 (0.42) CPB1FKBP1ATSHRALDH1A1CYP2C9
SCHEMBL8723700 0.71 ALDH1A1 (0.43) FKBP1ATSHRALDH1A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed