SCHEMBL6289334

SCHEMBL6289334

CN1C(=O)C(Cc2ccc(F)cc2)Cc2oc(C(=O)NCc3ccccc3)nc21

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
CACNA1G O43497 1/20 0.41
THRB P10828 1/20 0.41
CCR3 P51677 1/20 0.40
SCD O00767 1/20 0.40
CNR2 P34972 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6701897 0.80 SCD (0.52) ALDH1A1LMNAKDM4EHPGDSMN1; SMN2
SCHEMBL6289333 0.71 LMNA (0.44) ALDH1A1LMNAKDM4EHPGDSMN1; SMN2
SCHEMBL6288787 0.70 PTGER4 (0.46) ALDH1A1SCDMAPTTP53
SCHEMBL6292734 0.70 LMNA (0.47) ALDH1A1LMNAKDM4EHPGDSMN1; SMN2
SCHEMBL6748396 0.69 SMN1; SMN2 (0.43) ALDH1A1LMNASMN1; SMN2KMT2AMEN1
SCHEMBL6288765 0.68 HPGD (0.47) ALDH1A1LMNAKDM4EHPGDSMN1; SMN2
SCHEMBL6292798 0.67 PTGER4 (0.40) ALDH1A1LMNAKDM4EHPGDSMN1; SMN2
SCHEMBL6745755 0.66 MAPT (0.47) LMNASMN1; SMN2THRBMAPTTP53
SCHEMBL17804027 0.66 SCD (0.45) ALDH1A1LMNASMN1; SMN2THRBCCR3
SCHEMBL3043662 0.66 SCD (0.66) SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6949651-B2 Fused bicyclic metalloproteinase inhibitors WARNER-LAMBERT COMPANY (US) 2005-09-27 US disclosed
US-20040034054-A1 Fused bicyclic metalloproteinase inhibitors LINCOLN FOODSERVICE PRODUCTS INC. 2004-02-19 US disclosed
WO-2004014375-A2 FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034054-A1 Fused bicyclic metalloproteinase inhibitors MMP9, MMP1, MMP2 ALDH1A1 337/4885LMNA 1817/4885KDM4E 1792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.