SCHEMBL6293241

SCHEMBL6293241

CN(C)CC1CCC(=O)C=C1c1cccc(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
CCR6 P51684 1/20 0.40
METAP1 P53582 3/20 0.31
BACE1 P56817 1/20 0.31
HTR6 P50406 4/20 0.31
NCOA1 Q15788 1/20 0.30
NCOA3 Q9Y6Q9 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
SLC16A3 O15427 1/20 0.30
SLC16A1 P53985 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7595498 0.82 HSP90AA1 (0.52) HSP90AA1CCR6METAP1HTR6NCOA1
Hydrochloric Acid SCHEMBL6293297 0.82 HSP90AA1 (0.57) HSP90AA1CCR6METAP1HTR6NCOA1
SCHEMBL2969421 0.81 HSP90AA1 (0.55) HSP90AA1CCR6METAP1HTR6NCOA1
SCHEMBL6293028 0.77 METAP1 (0.41) HSP90AA1CCR6METAP1HTR6
SCHEMBL6294309 0.73 SLC6A3 (0.40) HSP90AA1CCR6METAP1HTR6
SCHEMBL6294523 0.73 HSP90AA1 (0.40) HSP90AA1CCR6HTR6
SCHEMBL6298674 0.73 ADRA2A (0.41) HSP90AA1CCR6
SCHEMBL6298643 0.71 HSP90AA1 (0.38) HSP90AA1CCR6METAP1HTR6
SCHEMBL6681699 0.70 HSP90AA1 (0.47) HSP90AA1CCR6METAP1HTR6
SCHEMBL6297691 0.69 METAP1 (0.45) HSP90AA1CCR6METAP1BACE1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890959-B2 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2005-05-10 US disclosed
EP-1246791-B1 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES GRUENENTHAL GMBH (DE) 2004-10-27 EP disclosed
US-20030096811-A1 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2003-05-22 US disclosed
EP-1246791-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2002-10-09 EP disclosed
WO-2001049651-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2001-07-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030096811-A1 Aminomethyl-phenyl-cyclohexanone derivatives CYP2J2, CYP2E1, CYP2D6 HSP90AA1 1369/4885CCR6 970/4885METAP1 1551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.