SCHEMBL6298643

SCHEMBL6298643

CN(C)CC1CCC(=O)C=C1c1cccc(C(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.38
CCR6 P51684 1/20 0.38
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
GRIN2B Q13224 4/20 0.35
GRIN1 Q05586 2/20 0.35
NOTUM Q6P988 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
METAP1 P53582 2/20 0.32
HTR6 P50406 1/20 0.32
MITF O75030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6294523 0.84 HSP90AA1 (0.40) HSP90AA1CCR6ADRA2AADRA2BADRA2C
SCHEMBL6298674 0.81 ADRA2A (0.41) HSP90AA1CCR6ADRA2AADRA2BADRA2C
SCHEMBL6293028 0.81 METAP1 (0.41) HSP90AA1CCR6ADRA2AADRA2BADRA2C
SCHEMBL2969421 0.81 HSP90AA1 (0.55) HSP90AA1CCR6BRD4METAP1HTR6
Hydrochloric Acid SCHEMBL6293297 0.80 HSP90AA1 (0.57) HSP90AA1CCR6BRD4METAP1HTR6
SCHEMBL7595498 0.78 HSP90AA1 (0.52) HSP90AA1CCR6BRD4METAP1HTR6
SCHEMBL6294319 0.78 HSP90AA1 (0.36) HSP90AA1CCR6ADRA2AADRA2BADRA2C
SCHEMBL6294309 0.77 SLC6A3 (0.40) HSP90AA1CCR6METAP1HTR6
SCHEMBL6294496 0.76 HSP90AA1 (0.36) HSP90AA1CCR6ADRA2AADRA2BADRA2C
SCHEMBL6297665 0.76 HSP90AA1 (0.35) HSP90AA1CCR6ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890959-B2 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2005-05-10 US claimed
EP-1246791-B1 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES GRUENENTHAL GMBH (DE) 2004-10-27 EP claimed
US-20030096811-A1 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2003-05-22 US claimed
EP-1246791-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2002-10-09 EP claimed
WO-2001049651-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2001-07-12 WO claimed
US-6890959-B2 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2005-05-10 US disclosed
EP-1246791-B1 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES GRUENENTHAL GMBH (DE) 2004-10-27 EP disclosed
US-20030096811-A1 Aminomethyl-phenyl-cyclohexanone derivatives GRUENENTHAL GMBH (DE) 2003-05-22 US disclosed
EP-1246791-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2002-10-09 EP disclosed
WO-2001049651-A2 AMINOMETHYL-PHENYL-CYCLOHEXANONE DERIVATIVES Grünenthal GmbH (DE) 2001-07-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030096811-A1 Aminomethyl-phenyl-cyclohexanone derivatives CYP2J2, CYP2E1, CYP2D6 HSP90AA1 1369/4885CCR6 970/4885BRD4 4043/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.