SCHEMBL6299196

SCHEMBL6299196

Cc1sc2ccc(C(=O)O)cc2c1Cc1cccc(Cl)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TBXAS1 P24557 2/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PFKFB4 Q16877 2/20 0.38
PFKFB3 Q16875 1/20 0.38
NR4A2 P43354 1/20 0.38
TTR P02766 2/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PTGER4 P35408 1/20 0.36
PTGER2 P43116 1/20 0.36
PTPRC P08575 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300210 0.91 SLC22A12 (0.42) SLC22A12SMN1; SMN2TBXAS1NPC1RAB9A
SCHEMBL6301947 0.89 MAPT (0.43) SLC22A12MEN1KMT2APFKFB4PFKFB3
SCHEMBL6299012 0.82 NR4A2 (0.44) SMN1; SMN2TBXAS1NPC1RAB9APFKFB4
SCHEMBL6300093 0.82 MRGPRX4 (0.40) SMN1; SMN2TBXAS1NPC1RAB9APFKFB4
SCHEMBL6298858 0.81 ACLY (0.38) SMN1; SMN2TBXAS1MRGPRX4ALDH1A1HPGD
SCHEMBL6299476 0.81 PTGER4 (0.39) SLC22A12SMN1; SMN2TBXAS1NPC1RAB9A
SCHEMBL6305986 0.81 ALDH1A1 (0.40) SLC22A12SMN1; SMN2TBXAS1NPC1RAB9A
SCHEMBL6301214 0.81 PDE3B (0.47) SLC22A12SMN1; SMN2NPC1RAB9APFKFB4
SCHEMBL6299126 0.79 TBXAS1 (0.48) SMN1; SMN2TBXAS1NPC1RAB9AALDH1A1
SCHEMBL6306599 0.79 TSHR (0.45) SMN1; SMN2TBXAS1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911469-B2 Sulfonamide compounds and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-28 US disclosed
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-09-16 US disclosed
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2002-07-25 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-0995742-A1 SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity PDE2A, PDE3A, PDE12 SLC22A12 822/4885SMN1; SMN2 186/4885NPSR1 463/4885
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications PDE2A, PDE3A, PYGM SLC22A12 1685/4885SMN1; SMN2 1017/4885NPSR1 1699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.