SCHEMBL6300922

SCHEMBL6300922

CCCC(=O)N(C)c1cc[c]c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.37
NPY5R Q15761 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 3/20 0.33
RAB9A P51151 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MCHR1 Q99705 1/20 0.32
AGPAT2 O15120 1/20 0.31
THRB P10828 1/20 0.31
POLQ O75417 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
EGFR P00533 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27556247 0.91 ALDH1A1 (0.40) ALDH1A1THRBHTT
SCHEMBL6135389 0.81 LMNA (0.45) ALDH1A1RAB9AHSD17B10MAPTMAPK1
SCHEMBL28687075 0.77 TP53 (0.43) TP53KDM4EALDH1A1RAB9AHSD17B10
SCHEMBL15979067 0.75 HTR3E (0.53) TP53KDM4EALDH1A1RAB9APOLQ
SCHEMBL6494236 0.75 NPY2R (0.41) CYP3A4
SCHEMBL22170065 0.74 DRD4 (0.44) TP53ALDH1A1RAB9AHSD17B10POLQ
SCHEMBL6299187 0.73 KMT2A (0.46) KDM4EALDH1A1RAB9AEGFRMAPT
SCHEMBL4011698 0.72 DAO (0.31)
SCHEMBL4006254 0.72 IGLV6-57 (0.34)
SCHEMBL6505131 0.72 LMNA (0.45) MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911469-B2 Sulfonamide compounds and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-28 US disclosed
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-09-16 US disclosed
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2002-07-25 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020099212-A1 For therapy of disease treatable based on a blood sugar level-depressing activity or a disease treatable based on a cGMP-PDE inhibiting activity, smooth muscle relaxing activity, bronchodilating activity, vasodilating activity PDE2A, PDE3A, PDE12 TP53 4884/4885NPY5R 393/4885KDM4E 1305/4885
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications PDE2A, PDE3A, PYGM TP53 4849/4885NPY5R 546/4885KDM4E 935/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.